SCHEMBL7040229

SCHEMBL7040229

NCCc1ccccc1-c1cccs1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.57
TAAR1 Q96RJ0 8/20 0.47
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46
ADRA2C P18825 1/20 0.41
HTR2A P28223 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ATM Q13315 1/20 0.39
TDO2 P48775 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HRH1 P35367 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3780733 0.85 LTA4H (0.61) LTA4HNPC1RAB9AATMTDO2
Hydrochloric Acid SCHEMBL2463750 0.83 LTA4H (0.59) LTA4HNPC1RAB9AATMTDO2
SCHEMBL3906600 0.81 LTA4H (0.57) LTA4HNPC1RAB9AATMTDO2
SCHEMBL3345523 0.80 LTA4H (0.56) LTA4HTAAR1NPC1RAB9AKDM4E
SCHEMBL5925309 0.79 LTA4H (0.54) LTA4HNPC1RAB9AATMKDM4E
SCHEMBL15244880 0.79 TAAR1 (0.48) TAAR1ADRA2CHTR2ASMN1; SMN2HRH1
SCHEMBL5925318 0.77 LTA4H (0.53) LTA4HNPC1RAB9AATMKDM4E
SCHEMBL5023959 0.77 LTA4H (0.66) LTA4HNPC1RAB9AKDM4EALDH1A1
SCHEMBL6028964 0.77 LTA4H (0.61) LTA4HNPC1RAB9AATMTDO2
SCHEMBL4846964 0.77 LTA4H (0.61) LTA4HNPC1RAB9AATMTDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0659737-B1 Catecholamine surrogates useful as beta 3 agonists BRISTOL MYERS SQUIBB CO (US) 2003-03-26 EP disclosed
US-5776983-A ANTIDIABETIC AGENTS, OBESITY, GASTROINTESTINAL DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-07-07 US disclosed
EP-0557305-B1 (2-THIENYL) ALKYLAMINE DERIVATIVES HAVING NEUROPROTECTIVE PROPERTIES ASTRA AB (SE) 1997-06-11 EP disclosed
EP-0659737-A2 Catecholamine surrogates useful as B3 agonists BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-28 EP disclosed
EP-0172692-B1 HEXAHYDROINDOLIZINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS AND INTERMEDIATES McNeilab, Inc. (US) 1990-04-18 EP disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed
EP-0172692-A1 Hexahydroindolizine compounds, pharmaceutical compositions and methods and intermediates McNeilab, Inc. (US) 1986-02-26 EP disclosed
US-4572911-A ANTISECRETORY AND ANTIDEPRESSANT AGENTS MCNEILAB, INC. (US) 1986-02-25 US disclosed