SCHEMBL7042363

SCHEMBL7042363

O=C(O)C(=O)c1cc(Br)sc1Br

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
CES2 O00748 2/20 0.35
CES1 P23141 2/20 0.35
DAO P14920 1/20 0.34
GSK3B P49841 2/20 0.34
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623602 0.82 TSHR (0.45) ALDH1A1CES2CES1DAOGSK3B
Hydrochloric Acid SCHEMBL29045760 0.80 TSHR (0.43) ALDH1A1DAOGSK3BTSHRKMT2A
SCHEMBL11841036 0.79 GSK3B (0.38) ALDH1A1CES2CES1DAOGSK3B
SCHEMBL28713332 0.76 GSK3B (0.35) ALDH1A1CES2CES1DAOGSK3B
SCHEMBL29114725 0.76 DGAT1 (0.39) ALDH1A1CES2CES1GSK3BTSHR
SCHEMBL7043307 0.72 MAPT (0.41) ALDH1A1TSHRKMT2A
SCHEMBL24198763 0.71 GSK3B (0.32) ALDH1A1GSK3B
SCHEMBL21054378 0.71 CA12 (0.40) ALDH1A1TSHRKMT2A
SCHEMBL3841520 0.71 ALDH1A1 (0.44) ALDH1A1GSK3BKMT2A
SCHEMBL7042303 0.70 GSK3B (0.57) CES2CES1DAOGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613786-B2 Treating urinary incontinence, asthma, irritable bowel syndrome or male erectile dysfunction BRISTOL-MYERS SQUIBB COMPANY 2003-09-02 US disclosed
US-20030144333-A1 Thiophenyl triazol-3-one derivatives as smooth muscle relaxants HEWAWASAM PIYASENA (US) 2003-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030144333-A1 Thiophenyl triazol-3-one derivatives as smooth muscle relaxants PDE3A, ADRB2, ADRB3 ALDH1A1 1237/4885CES2 2835/4885CES1 945/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.