SCHEMBL7042941

SCHEMBL7042941

CSC(=O)Cc1ccc(C(=O)N(C)C)c(Cl)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
HPGD P15428 2/20 0.35
HTT P42858 1/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 2/20 0.33
POLB P06746 1/20 0.33
THRB P10828 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PDK2 Q15119 1/20 0.30
THRA P10827 1/20 0.30
MAP4K1 Q92918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5208590 0.75 ALDH1A1 (0.42) ALDH1A1HPGDHTTMEN1KMT2A
SCHEMBL6136980 0.69 CXCL8 (0.36) ALDH1A1MAPT
SCHEMBL23021682 0.68 ALDH1A1 (0.51) ALDH1A1HPGDHTTMEN1KMT2A
SCHEMBL3791684 0.67 SMN1; SMN2 (0.52) ALDH1A1HPGDHTTMEN1KMT2A
SCHEMBL19286776 0.65 CTBP2 (0.50) ALDH1A1HTTKMT2AMAPTSMN1; SMN2
SCHEMBL23021795 0.61 ALDH1A1 (0.47) ALDH1A1HPGDHTTMEN1KMT2A
SCHEMBL15434614 0.60 GABRA1 (0.41) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL3780795 0.60 HPGD (0.58) ALDH1A1HPGDHTTMEN1KMT2A
SCHEMBL27308477 0.60 CLCN2 (0.54) ALDH1A1HPGDMEN1KMT2AMAPT
SCHEMBL18931210 0.60 ALDH1A1 (0.50) ALDH1A1HPGDHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882029-B1 HETEROCYCLIC DERIVATIVES AS ANTIDIABETIC AND ANTIOBESITY AGENTS MERCK & CO INC (US) 2003-04-02 EP disclosed
US-6090836-A DIETETICS; ADJUSTMENT OF TRIGLYCERIDE CONCENTRATION MERCK & CO., INC. (US) 2000-07-18 US disclosed
EP-0882029-A1 HETEROCYCLIC DERIVATIVES AS ANTIDIABETIC AND ANTIOBESITY AGENTS Merck & Co., Inc. (US) 1998-12-09 EP disclosed
WO-1997028137-A1 HETEROCYCLIC DERIVATIVES AS ANTIDIABETIC AND ANTIOBESITY AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed