SCHEMBL7043751

SCHEMBL7043751

Cn1c(N2CCCN(CCc3ccc(Cl)cc3)CC2)nc2c(OC(N)=O)cccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.39
DRD3 P35462 2/20 0.39
HTR2A P28223 2/20 0.39
HRH1 P35367 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
HTR1A P08908 1/20 0.39
HTR2C P28335 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
THRB P10828 1/20 0.38
ABCC1 P33527 3/20 0.38
CYP3A4 P08684 1/20 0.38
DRD4 P21917 2/20 0.38
SMYD2 Q9NRG4 2/20 0.37
GRM2 Q14416 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7044886 0.96 THRB (0.41) DRD2HTR2ASIGMAR1THRBABCC1
SCHEMBL7038533 0.88 PARP1 (0.47) DRD2NPSR1PARP1
SCHEMBL5619701 0.86 PARP1 (0.51) DRD2ABCC1CYP3A4DRD4GRM2
SCHEMBL7040971 0.85 HTR7 (0.42) DRD2DRD3HTR1ACYP3A4DRD4
SCHEMBL7039979 0.84 PARP1 (0.50) DRD2SIGMAR1KDM4EMEN1GAA
SCHEMBL7042531 0.83 PARP1 (0.56) DRD2DRD3HTR2AHRH1CYP3A4
SCHEMBL5621817 0.82 PARP1 (0.54) DRD2HTR2ASIGMAR1ABCC1CYP3A4
SCHEMBL6864807 0.81 PARP1 (0.40) DRD2DRD3HTR2AHRH1SIGMAR1
SCHEMBL7038527 0.81 PARP1 (0.52) DRD3HRH1DRD4MEN1KMT2A
SCHEMBL7041477 0.81 DRD2 (0.44) DRD2DRD3HTR1ADRD4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed