SCHEMBL7046067

SCHEMBL7046067

O=C(O)Nc1nc2cc(S(=O)(=O)Cl)ccc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.43
RAB9A P51151 7/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
PKM P14618 2/20 0.43
MAOB P27338 1/20 0.43
ADORA2A P29274 1/20 0.43
POLB P06746 1/20 0.42
KDM4E B2RXH2 2/20 0.42
LMNA P02545 2/20 0.42
HTT P42858 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ALDH1A1 P00352 3/20 0.42
CYP3A4 P08684 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPK1 P28482 2/20 0.40
HSD17B10 Q99714 2/20 0.40
SCD O00767 1/20 0.39
OPRK1 P41145 1/20 0.39
KLF5 Q13887 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4862487 0.85 ACR (0.52) NPC1SMN1; SMN2ADORA2AKDM4ELMNA
SCHEMBL10896181 0.85 NPC1 (0.48) NPC1RAB9ASMN1; SMN2PKMMAOB
Hydrochloric Acid SCHEMBL10732492 0.84 ACR (0.51) NPC1SMN1; SMN2ADORA2AKDM4ELMNA
SCHEMBL11095372 0.84 TUBB4A (0.45) SMN1; SMN2POLBLMNAHTTMEN1
Hydrochloric Acid SCHEMBL11094572 0.83 TUBB4A (0.44) SMN1; SMN2POLBLMNAHTTMEN1
SCHEMBL28209330 0.81 IRAK4 (0.53) NPC1RAB9ASMN1; SMN2PKMKDM4E
SCHEMBL11524230 0.81 SMN1; SMN2 (0.41) NPC1RAB9ASMN1; SMN2PKMMAOB
SCHEMBL4865913 0.79 NPSR1 (0.46) NPC1RAB9ASMN1; SMN2POLBKDM4E
SCHEMBL9719979 0.78 NPC1 (0.54) NPC1RAB9ASMN1; SMN2PKMMAOB
SCHEMBL4637243 0.78 NPC1 (0.48) NPC1RAB9ASMN1; SMN2PKMMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1485358-A1 BROADSPECTRUM SUBSTITUTED BENZIMIDAZOLE SULFONAMIDE HIV PROTEASE INHIBITORS Tibotec Pharmaceuticals Ltd. (IE) 2004-12-15 EP disclosed
WO-2003076413-A1 BROADSPECTRUM SUBSTITUTED BENZIMIDAZOLE SULFONAMIDE HIV PROTEASE INHIBITORS TIBOTEC PHARMACEUTICALS LTD (IE) 2003-09-18 WO disclosed