SCHEMBL7046455

SCHEMBL7046455

CCCCCCN(C)C(=O)c1nc(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2)[nH]1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CNR1 P21554 2/20 0.44
GCGR P47871 1/20 0.43
HRH4 Q9H3N8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7048218 0.90
SCHEMBL7046399 0.89 CNR1 (0.51) KDM4EALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL7044567 0.88 CSNK2A2 (0.47)
SCHEMBL7046656 0.87 CNR1 (0.52) KDM4EALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL7044710 0.80 KDM4E (0.43) KDM4EALDH1A1HPGDSMN1; SMN2CNR1
SCHEMBL7041234 0.77 CNR1 (0.48) KDM4EALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL7046157 0.76 CNR1 (0.49) CNR1GCGR
SCHEMBL5268736 0.72 CNR1 (0.58) KDM4EALDH1A1HPGDCNR1GCGR
SCHEMBL7043396 0.71 CNR1 (0.61) ALDH1A1HPGDCNR1
SCHEMBL7046592 0.71 CNR1 (0.61) CNR1GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007887-A2 SUBSTITUTED IMIDAZOLES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-01-30 WO claimed
WO-2003007887-A2 SUBSTITUTED IMIDAZOLES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-01-30 WO disclosed