SCHEMBL7046578

SCHEMBL7046578

CCCC1(CCC)CCCNC1=O

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
CYP19A1 P11511 4/20 0.35
HSD11B1 P28845 7/20 0.33
CYP2D6 P10635 3/20 0.31
SLC6A2 P23975 3/20 0.31
SLC6A4 P31645 3/20 0.31
SLC6A3 Q01959 3/20 0.31
KCNH2 Q12809 1/20 0.31
CCR2 P41597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19534246 0.88 CYP19A1 (0.40) CYP19A1HSD11B1
SCHEMBL6730153 0.83 GRIN1 (0.38) GRIN1GRIN2ACYP19A1HSD11B1
SCHEMBL28358676 0.82 CYP19A1 (0.43) CYP19A1CCR2
SCHEMBL11196121 0.77 CYP19A1 (0.36) GRIN1GRIN2ACYP19A1HSD11B1CYP2D6
SCHEMBL3272687 0.74 GRIN1 (0.33) GRIN1GRIN2A
SCHEMBL21585193 0.74 POLB (0.36) CYP19A1HSD11B1
SCHEMBL14378012 0.73 MMP9 (0.33) GRIN1GRIN2ACCR2
SCHEMBL22213505 0.72 CYP19A1 (0.38) GRIN1GRIN2ACYP19A1CCR2
SCHEMBL28870336 0.72 CCR2 (0.33) GRIN1GRIN2ACYP19A1CCR2
SCHEMBL9800283 0.71 GRIN1 (0.33) GRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007940-A1 LACTAM AND THIOLACTAM DERIVATIVES AS ANESTHETIC AND CONSCIOUS SEDATION AGENTS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2003-01-30 WO disclosed
US-5003082-A Reacting a lactam with hydrogen sulfide in the presence of an inorganic catalyst PHILLIPS PETROLEUM COMPANY (US) 1991-03-26 US disclosed
US-4990628-A Reacting lactam with hydrogen sulfide in presence of group 8 metals or compounds on alumina; support; sulfiding PHILLIPS PETROLEUM COMPANY (US) 1991-02-05 US disclosed
US-4956476-A Catalytic reaction of a lactam with hydrogen sulfide to produce a thiolactam, alumina is the catalyst PHILLIPS PETROLEUM COMPANY (US) 1990-09-11 US disclosed
US-4145352-A SULFACTIVE CATALYST PHILLIPS PETROLEUM COMPANY (US) 1979-03-20 US disclosed