SCHEMBL7048567

SCHEMBL7048567

COc1cc(C#N)ccc1CNC(=O)OC1CCN1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.46
JAK1 P23458 1/20 0.46
TYK2 P29597 1/20 0.46
JAK3 P52333 1/20 0.46
HPGD P15428 2/20 0.41
ENPP2 Q13822 1/20 0.41
HTR2A P28223 2/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
P2RX7 Q99572 1/20 0.39
IDH1 O75874 1/20 0.38
DRD2 P14416 2/20 0.38
DRD1 P21728 2/20 0.38
DRD4 P21917 2/20 0.38
DRD5 P21918 2/20 0.38
DRD3 P35462 2/20 0.38
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6483702 0.81 HTR2C (0.59) JAK2JAK1TYK2JAK3HPGD
SCHEMBL6483706 0.81 HTR2C (0.59) JAK2JAK1TYK2JAK3HPGD
Hydrochloric Acid SCHEMBL7044040 0.80 HTR2C (0.58) JAK2JAK1TYK2JAK3HPGD
Hydrochloric Acid SCHEMBL8377589 0.80 HTR2C (0.58) JAK2JAK1TYK2JAK3HPGD
SCHEMBL23755099 0.79 SETDB1 (0.44) JAK2JAK1TYK2JAK3ENPP2
SCHEMBL30791546 0.79 SETDB1 (0.53) JAK2JAK1TYK2JAK3ENPP2
SCHEMBL30305200 0.79 ABCB1 (0.43) JAK2JAK1TYK2JAK3ENPP2
SCHEMBL23775495 0.79 ABCB1 (0.43) JAK2JAK1TYK2JAK3ENPP2
SCHEMBL7050773 0.77 ALDH1A1 (0.42) JAK2JAK1TYK2JAK3HPGD
SCHEMBL29196350 0.73 HTR2A (0.47) HTR2AIDH1ALDH1A1KCNH2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773955-B1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AG (DE) 2003-04-16 EP disclosed
EP-0773955-A1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1997-05-21 EP disclosed
WO-1995035309-A1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1995-12-28 WO disclosed