SCHEMBL7050773

SCHEMBL7050773

COc1cc(C#N)ccc1CNC(=O)OC1CCN1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
JAK3 P52333 1/20 0.41
EPHX2 P34913 1/20 0.41
KDM4D Q6B0I6 1/20 0.41
GPR119 Q8TDV5 3/20 0.39
DRD2 P14416 2/20 0.39
ENPP2 Q13822 1/20 0.39
HPGD P15428 2/20 0.36
NSD2 O96028 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7047070 0.83 ALDH1A1 (0.64) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL23775495 0.81 ABCB1 (0.43) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL30305200 0.81 ABCB1 (0.43) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL7048567 0.77 JAK2 (0.46) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL30924101 0.72 EPHX2 (0.59) EPHX2GPR119
SCHEMBL7046882 0.71 JAK2 (0.39) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL30791546 0.71 SETDB1 (0.53) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL23755099 0.71 SETDB1 (0.44) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL7050252 0.70 ALDH1A1 (0.79) ALDH1A1
SCHEMBL24837810 0.70 TRPV1 (0.42) ALDH1A1DRD2HPGDTSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773955-B1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AG (DE) 2003-04-16 EP disclosed
WO-1995035309-A1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1995-12-28 WO disclosed