SCHEMBL7049656

SCHEMBL7049656

C=Cc1c(C)cc(N)nc1C

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 12/20 0.40
NOS3 P29474 8/20 0.40
NOS1 P29475 7/20 0.40
BACE1 P56817 1/20 0.37
REN P00797 1/20 0.36
PRMT5 O14744 1/20 0.34
KLKB1 P03952 1/20 0.30
PDXK O00764 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31256111 0.80 NOS2 (0.34) NOS2NOS3NOS1
SCHEMBL8328225 0.79 BACE1 (0.41) NOS2NOS3NOS1BACE1REN
SCHEMBL20663167 0.77 NOS2 (0.33) NOS2NOS3NOS1BACE1PRMT5
SCHEMBL26660403 0.76 BACE1 (0.44) NOS2NOS3NOS1BACE1
SCHEMBL7115996 0.75 PDXK (0.30) PDXK
SCHEMBL21632441 0.71 NOS2 (0.44) NOS2NOS3NOS1BACE1REN
SCHEMBL3673476 0.70 NOS2 (0.48) NOS2NOS3NOS1BACE1REN
SCHEMBL5758060 0.70 NOS2 (0.48) NOS2NOS3NOS1BACE1REN
SCHEMBL9284246 0.70 KDM4E (0.40) PDXK
SCHEMBL31256219 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972975-A Substituted 2-aminopyridines as inhibitors of nitric oxide synthase MERCK & CO., INC. (US) 1999-10-26 US claimed
WO-1996018616-A1 SUBSTITUTED 2-AMINOPYRIDINES AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO., INC. (US) 1996-06-20 WO claimed
CN-108950645-B Aluminum and aluminum alloy anodic oxidation nickel-free sealing agent 上海铝通化学科技有限公司 2020-10-23 CN disclosed
WO-2003013523-A1 SH3 PROTEIN DOMAINS AND THEIR LIGANDS ADELAIDE RESEARCH & INNOVATION PTY LTD (AU) 2003-02-20 WO disclosed
US-5972975-A Substituted 2-aminopyridines as inhibitors of nitric oxide synthase MERCK & CO., INC. (US) 1999-10-26 US disclosed
WO-1996018616-A1 SUBSTITUTED 2-AMINOPYRIDINES AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO., INC. (US) 1996-06-20 WO disclosed