Bromide

Bromide

SCHEMBL7050720

Cc1sc[n+](CC(=O)N2C(C)CCCC2C)c1C.Cc1sc[n+](CC(=O)N2CCCCC2C)c1C.Cc1sc[n+](CC(=O)N2CCCCCCC2)c1C.Cc1sc[n+](CC(=O)c2ccccn2)c1C.[Br-].[Br-].[Cl-].[Cl-]

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
RAB9A P51151 4/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
ATM Q13315 1/20 0.36
KMT2A Q03164 4/20 0.35
TRPC3 Q13507 1/20 0.35
TRPC6 Q9Y210 1/20 0.35
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 1/20 0.34
LMNA P02545 2/20 0.34
TP53 P04637 2/20 0.34
HPGD P15428 2/20 0.33
NPC1 O15118 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL5978880 0.96 ALDH1A1 (0.38) ALDH1A1RAB9AMAPTMAPK1ATM
Bromide SCHEMBL6425488 0.88 SMN1; SMN2 (0.36) ALDH1A1MAPK1KMT2AKDM4ETP53
Bromide SCHEMBL5015757 0.87 KMT2A (0.44) ALDH1A1RAB9AMAPTKMT2AKDM4E
SCHEMBL6772875 0.81 ALDH1A1 (0.38) ALDH1A1RAB9AMAPTMAPK1ATM
Hydrochloric Acid SCHEMBL3848955 0.80 HPGD (0.44) ALDH1A1RAB9AMAPK1ATMKMT2A
SCHEMBL5071288 0.79 HPGD (0.45) ALDH1A1RAB9AMAPK1ATMKMT2A
Bromide SCHEMBL7052826 0.77 ALDH1A1 (0.33) ALDH1A1RAB9AMAPTMAPK1ATM
Hydrochloric Acid SCHEMBL3847184 0.77 HPGD (0.43) ALDH1A1RAB9AMAPTATMKMT2A
Bromide SCHEMBL8081586 0.77 KMT2A (0.54) ALDH1A1RAB9AKMT2ALMNANPC1
Bromide SCHEMBL3843812 0.77 KMT2A (0.54) ALDH1A1RAB9AKMT2ALMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1128830-A4 REVERSING ADVANCED GLYCOSYLATION CROSS-LINKS USING HETEROCYCLIC-SUBSTITUTED THIAZOLIUM SALTS ALTEON INC (US) 2004-03-31 EP disclosed
EP-1128830-A1 REVERSING ADVANCED GLYCOSYLATION CROSS-LINKS USING HETEROCYCLIC-SUBSTITUTED THIAZOLIUM SALTS Alteon, Inc. (US) 2001-09-05 EP disclosed
WO-2000027395-A1 REVERSING ADVANCED GLYCOSYLATION CROSS-LINKS USING HETEROCYCLIC-SUBSTITUTED THIAZOLIUM SALTS ALTEON, INC. (US) 2000-05-18 WO disclosed