SCHEMBL7051878

SCHEMBL7051878

CCn1cc(C(=O)NCCc2cccnc2)c(=O)c2cccc(C(F)(F)F)c21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 7/20 0.53
PDE4B Q07343 7/20 0.53
PDE4C Q08493 7/20 0.53
PDE4D Q08499 7/20 0.53
ALDH1A1 P00352 5/20 0.47
KDM4E B2RXH2 3/20 0.47
MAPK1 P28482 1/20 0.47
PDE10A Q9Y233 1/20 0.47
CNR2 P34972 2/20 0.47
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
HPGD P15428 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CACNA1B Q00975 1/20 0.43
APBA1 Q02410 1/20 0.43
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7056153 0.92 ALDH1A1 (0.56) ALDH1A1KDM4EMAPK1PDE10AMEN1
SCHEMBL7051834 0.89 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7057844 0.84 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7054222 0.83 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7057001 0.83 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7055521 0.83 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7058521 0.83 CNR2 (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7050618 0.83 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7055640 0.81 LMNA (0.58) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7051841 0.81 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0841929-B1 QUINOLONES AND THEIR THERAPEUTIC USE DARWIN DISCOVERY LTD (GB) 2003-05-07 EP claimed