SCHEMBL7051943

SCHEMBL7051943

O=C(CCF)N1CCN(c2ncnc3sc(-c4ccccc4)cc23)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.72
ALDH1A1 P00352 10/20 0.72
MAPT P10636 4/20 0.64
POLB P06746 3/20 0.64
RXFP1 Q9HBX9 2/20 0.64
LMNA P02545 1/20 0.64
GAA P10253 3/20 0.64
MEN1 O00255 5/20 0.63
SMN1; SMN2 Q16637 4/20 0.63
KMT2A Q03164 3/20 0.63
MAPK1 P28482 4/20 0.63
NPSR1 Q6W5P4 2/20 0.61
MCL1 Q07820 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
PKM P14618 1/20 0.61
HPGD P15428 2/20 0.60
HSD17B10 Q99714 2/20 0.60
USP2 O75604 1/20 0.60
P2RY12 Q9H244 5/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5849667 0.87 KDM4E (0.71) KDM4EALDH1A1MAPTPOLBRXFP1
SCHEMBL5848988 0.87 ALDH1A1 (0.74) KDM4EALDH1A1MAPTPOLBRXFP1
SCHEMBL7062128 0.86 KDM4E (0.83) KDM4EALDH1A1MAPTPOLBRXFP1
SCHEMBL7051947 0.82 KDM4E (0.76) KDM4EALDH1A1MAPTPOLBRXFP1
SCHEMBL14825132 0.79 KDM4E (1.00) KDM4EALDH1A1MAPTPOLBRXFP1
SCHEMBL5851429 0.79 KDM4E (0.74) KDM4EALDH1A1MAPTPOLBRXFP1
SCHEMBL5851312 0.79 KDM4E (0.56) KDM4EALDH1A1MAPTPOLBRXFP1
SCHEMBL5851314 0.78 KDM4E (0.56) KDM4EALDH1A1MAPTPOLBRXFP1
SCHEMBL5850858 0.74 P2RY12 (0.82) KDM4EALDH1A1MAPTLMNAMEN1
SCHEMBL16090496 0.74 P2RY12 (0.64) ALDH1A1MEN1KMT2AP2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003022214-A2 PIPERAZINE AND HOMOPIPERAZINE COMPOUNDS MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-03-20 WO disclosed