SCHEMBL7051954

SCHEMBL7051954

COCCNC(=O)COc1ccc(C2CCC(CNC[C@H](O)c3cccc(Cl)c3)C2)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 15/20 0.46
ADRB1 P08588 12/20 0.46
ADRB2 P07550 5/20 0.45
GLA P06280 1/20 0.44
CYP2D6 P10635 3/20 0.43
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7051952 1.00 ADRB3 (0.46) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL7059933 0.88 ADRB3 (0.49) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL7059932 0.88 ADRB3 (0.49) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL7059103 0.85 ADRB3 (0.49) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL7059105 0.85 ADRB3 (0.49) ADRB3ADRB1ADRB2GLACYP2D6
Hydrochloric Acid SCHEMBL7054734 0.85 ADRB3 (0.59) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL7058088 0.83 ADRB3 (0.43) ADRB3ADRB1ADRB2GLA
Hydrochloric Acid SCHEMBL7057667 0.77 ADRB3 (0.45) ADRB3ADRB1ADRB2
SCHEMBL7051168 0.77 OPRK1 (0.46) ADRB3ADRB1ADRB2CYP3A4CYP2C9
SCHEMBL7051162 0.77 OPRK1 (0.46) ADRB3ADRB1ADRB2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0940387-B1 PHENYLETHANOLAMINE COMPOUNDS USEFUL AS BETA3 AGONIST, PROCESS FOR PRODUCING THE SAME, AND INTERMEDIATES IN THE PRODUCTION OF THE SAME MITSUBISHI PHARMA CORP (JP) 2003-05-07 EP disclosed
US-6069176-A PHENYLETHANOLAMINE COMPOUNDS WITH A BETA-3 ADRENERGIC RECEPTOR STIMULATING EFFECT, USE AS A THERAPY FOR URINARY INCONTINENCE MITSUBISHI-TOKYO PHARMACEUTICALS, INC. (JP) 2000-05-30 US disclosed
EP-0940387-A1 PHENYLETHANOLAMINE COMPOUNDS USEFUL AS BETA3 AGONIST, PROCESS FOR PRODUCING THE SAME, AND INTERMEDIATES IN THE PRODUCTION OF THE SAME TOKYO TANABE COMPANY LIMITED (JP) 1999-09-08 EP disclosed