SCHEMBL7052015

SCHEMBL7052015

O=C1CN(S(=O)(=O)c2ccc3cc(Cl)ccc3c2)CCN1C(c1cc(NCc2ccccc2)ncn1)C1(O)CCNCC1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
F10 P00742 13/20 0.37
MAPT P10636 2/20 0.37
TP53 P04637 1/20 0.37
F2 P00734 2/20 0.36
GCK P35557 1/20 0.34
PKM P14618 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7053488 0.86 F10 (0.40) F10F2GCKPKMSMN1; SMN2
SCHEMBL7052228 0.80 F10 (0.42) F10F2GCKPKM
Hydrochloric Acid SCHEMBL6888194 0.77 PIK3CB (0.38) TP53
SCHEMBL7052011 0.76 METTL3 (0.42) F10MAPTTP53F2
Hydrochloric Acid SCHEMBL7049914 0.68 F10 (0.44) F10MAPTF2PKMSMN1; SMN2
Hydrochloric Acid SCHEMBL5743404 0.64 F10 (0.39) F10MAPTF2
Hydrochloric Acid SCHEMBL7050611 0.64 F10 (0.41) F10F2
Hydrochloric Acid SCHEMBL7053310 0.63 F10 (0.41) F10MAPTF2PKM
Hydrochloric Acid SCHEMBL7050846 0.63 F10 (0.39) F10MAPTF2PKMSMN1; SMN2
SCHEMBL7053479 0.61 F10 (0.43) F10F2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6680312-B2 FOR THERAPY OF CARDIAC INFARCTION, CEREBRAL THROMBOSIS; INHIBIT ACTIVATED COAGULATION FACTOR X (FXA) TO SHOW ANTI-COAGULANT ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-01-20 US disclosed
US-20020193382-A1 Sulfonamide derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2002-12-19 US disclosed
US-6403595-B1 ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-06-11 US disclosed
EP-1054005-A1 SULFONAMIDE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-11-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020193382-A1 Sulfonamide derivatives, their production and use F12, F11, F2 F10 5/4885MAPT 4851/4885TP53 4755/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.