SCHEMBL7052959

SCHEMBL7052959

CNC(=O)Nc1sc(-c2ccc(O)c(OC)c2)cc1C(=O)NC

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 6/20 0.49
MAP4K4 O95819 1/20 0.49
HDAC6 Q9UBN7 1/20 0.48
IKBKB O14920 2/20 0.42
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
AURKB Q96GD4 2/20 0.39
PTPN1 P18031 1/20 0.38
NTRK1 P04629 1/20 0.37
YES1 P07947 1/20 0.37
MAPK1 P28482 1/20 0.37
SNCA P37840 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058543 0.95 CHEK1 (0.50) CHEK1MAP4K4HDAC6IKBKBHSD17B1
SCHEMBL7055165 0.91 CHEK1 (0.54) CHEK1MAP4K4IKBKBKDM4EALDH1A1
SCHEMBL7055235 0.83 CHEK1 (0.62) CHEK1MAP4K4HDAC6IKBKBKDM4E
SCHEMBL7059399 0.81 PTPN1 (0.53) CHEK1MAP4K4IKBKBKDM4EALDH1A1
SCHEMBL7055995 0.80 CHEK1 (0.62) CHEK1MAP4K4HDAC6IKBKBALDH1A1
SCHEMBL7058336 0.78 CHEK1 (0.66) CHEK1MAP4K4IKBKBKDM4EALDH1A1
SCHEMBL7055932 0.78 CHEK1 (0.59) CHEK1MAP4K4HDAC6IKBKBKDM4E
SCHEMBL7052328 0.77 CHEK1 (0.78) CHEK1MAP4K4IKBKBKDM4EMAPT
SCHEMBL7051467 0.76 CHEK1 (0.56) CHEK1MAP4K4IKBKBKDM4EMAPT
SCHEMBL7050462 0.74 CHEK1 (0.54) CHEK1MAP4K4HDAC6IKBKBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed