SCHEMBL7055165

SCHEMBL7055165

CNC(=O)Nc1sc(-c2ccc(OC)c(OC)c2)cc1C(=O)NC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 9/20 0.54
MAP4K4 O95819 1/20 0.54
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PTPN1 P18031 1/20 0.47
IKBKB O14920 2/20 0.46
BRD4 O60885 1/20 0.42
BRD9 Q9H8M2 1/20 0.42
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7052959 0.91 CHEK1 (0.49) CHEK1MAP4K4KDM4EALDH1A1HPGD
SCHEMBL7059399 0.90 PTPN1 (0.53) CHEK1MAP4K4KDM4EALDH1A1HPGD
SCHEMBL7058336 0.86 CHEK1 (0.66) CHEK1MAP4K4KDM4EALDH1A1HPGD
SCHEMBL7058543 0.86 CHEK1 (0.50) CHEK1MAP4K4KDM4EALDH1A1HPGD
SCHEMBL7055235 0.85 CHEK1 (0.62) CHEK1MAP4K4KDM4EALDH1A1HPGD
SCHEMBL7053757 0.81 PTPN1 (0.62) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL7055932 0.80 CHEK1 (0.59) CHEK1MAP4K4KDM4EALDH1A1HPGD
SCHEMBL7055995 0.80 CHEK1 (0.62) CHEK1MAP4K4ALDH1A1MAPTGAA
SCHEMBL7052328 0.79 CHEK1 (0.78) CHEK1MAP4K4KDM4EMAPTIKBKB
SCHEMBL7051467 0.78 CHEK1 (0.56) CHEK1MAP4K4KDM4EMAPTIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO claimed
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed