SCHEMBL7051467

SCHEMBL7051467

CNC(=O)Nc1sc(-c2ccc(CO)cc2)cc1C(=O)NC

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 12/20 0.56
MAP4K4 O95819 1/20 0.56
IKBKB O14920 2/20 0.49
ALOX15 P16050 1/20 0.43
NPC1 O15118 2/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
PTPN5 P54829 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7057068 0.90 NPC1 (0.51) CHEK1MAP4K4IKBKBNPC1MAPT
SCHEMBL7058742 0.89 IKBKB (0.64) CHEK1IKBKB
SCHEMBL7055932 0.84 CHEK1 (0.59) CHEK1MAP4K4IKBKBNPC1MAPT
SCHEMBL7055995 0.84 CHEK1 (0.62) CHEK1MAP4K4IKBKBALOX15NPC1
SCHEMBL7052328 0.84 CHEK1 (0.78) CHEK1MAP4K4IKBKBALOX15NPC1
SCHEMBL7055235 0.82 CHEK1 (0.62) CHEK1MAP4K4IKBKBNPC1MAPT
SCHEMBL7050462 0.78 CHEK1 (0.54) CHEK1MAP4K4IKBKBALOX15NPC1
SCHEMBL7055165 0.78 CHEK1 (0.54) CHEK1MAP4K4IKBKBMAPTKDM4E
SCHEMBL7058130 0.77 CHEK1 (0.59) CHEK1MAP4K4IKBKBALOX15NPC1
SCHEMBL7052959 0.76 CHEK1 (0.49) CHEK1MAP4K4IKBKBMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO claimed
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed