SCHEMBL7053668

SCHEMBL7053668

Cc1c(Br)ccc(N2CCN(CCCCN3C(=O)c4ccccc4C3=O)CC2)c1C

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.61
ALDH1A1 P00352 2/20 0.61
MEN1 O00255 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
ALOX12 P18054 1/20 0.61
ADRA1D P25100 1/20 0.61
HTR7 P34969 1/20 0.61
ADRA1A P35348 1/20 0.61
ADRA1B P35368 1/20 0.61
KMT2A Q03164 1/20 0.61
HIF1A Q16665 1/20 0.61
HSD17B10 Q99714 1/20 0.61
KDM4E B2RXH2 1/20 0.60
GLA P06280 1/20 0.60
HPGD P15428 1/20 0.60
DRD2 P14416 5/20 0.58
DRD3 P35462 5/20 0.58
DRD4 P21917 2/20 0.58
MAOB P27338 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058203 0.82 HTR1A (0.60) HTR1AALDH1A1MEN1CYP3A4CYP2D6
SCHEMBL13484830 0.81 HTR1A (0.71) HTR1AALDH1A1MEN1CYP3A4CYP2D6
SCHEMBL14028451 0.79 HTR1A (0.79) HTR1ADRD2DRD3MAOB
SCHEMBL10835924 0.79 DRD2 (0.71) HTR1AALDH1A1MEN1CYP3A4CYP2D6
SCHEMBL7052842 0.78 CYP2D6 (0.44) HTR1AALDH1A1MEN1CYP2D6KMT2A
SCHEMBL7056520 0.78 DRD2 (0.66) HTR1AALDH1A1MEN1CYP3A4CYP2D6
SCHEMBL7056493 0.77 HTR1A (0.76) HTR1AALDH1A1MEN1CYP3A4CYP2D6
SCHEMBL21802140 0.77 DRD2 (0.85) HTR1AALDH1A1MEN1CYP3A4CYP2D6
SCHEMBL21802088 0.76 DRD2 (0.83) HTR1AALDH1A1MEN1CYP3A4CYP2D6
SCHEMBL16406297 0.76 HTR1A (0.67) HTR1AALDH1A1MEN1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed