SCHEMBL7052842

SCHEMBL7052842

Cc1c(Br)ccc(N2CCN(CCCCN)CC2)c1C

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.44
SIGMAR1 Q99720 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
BRD4 O60885 1/20 0.39
BRD9 Q9H8M2 1/20 0.39
HTR1A P08908 2/20 0.39
KCNH2 Q12809 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7057953 0.79 ALDH1A1 (0.47) CYP2D6SIGMAR1HSD17B10ALDH1A1KDM4E
SCHEMBL3198516 0.78 ALDH1A1 (0.62) ALDH1A1KDM4EHTR1AMEN1KMT2A
SCHEMBL7053668 0.78 HTR1A (0.61) CYP2D6HSD17B10ALDH1A1KDM4EHTR1A
SCHEMBL3187557 0.75 MEN1 (0.51) ALDH1A1HTR1AKCNH2MEN1KMT2A
SCHEMBL3200107 0.75 ADRA1B (0.60) CYP2D6SIGMAR1ALDH1A1KDM4ELMNA
SCHEMBL7052673 0.74 ADRA1B (0.48) CYP2D6SIGMAR1HSD17B10ALDH1A1KDM4E
SCHEMBL5186020 0.74 KCNH2 (0.51) ALDH1A1HTR1AKCNH2MEN1KMT2A
SCHEMBL4249377 0.74 ALDH1A1 (0.63) CYP2D6ALDH1A1KDM4EHTR1AMEN1
SCHEMBL7055589 0.73 HTR1A (0.52) CYP2D6HSD17B10ALDH1A1HTR1AMEN1
Hydrochloric Acid SCHEMBL12099351 0.72 ALDH1A1 (0.62) CYP2D6ALDH1A1KDM4EHTR1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed