SCHEMBL7055819

SCHEMBL7055819

CCc1cc2c(N3CCN(C(C=O)c4ccccc4)CC3)nc(Cl)nc2s1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HTR6 P50406 1/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 3/20 0.46
P2RY12 Q9H244 15/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7046759 0.89 HTR6 (0.60) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL7051621 0.89 TP53 (0.47) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL7050247 0.89 P2RY12 (0.46) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL7047637 0.87 TP53 (0.45) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL7050374 0.87 TP53 (0.45) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL7055758 0.87 TP53 (0.45) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL7048623 0.84 HTT (0.67) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL7047651 0.78 HTT (0.45) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL7053533 0.77 HTT (0.56) TP53MAPTTSHRHTTSMN1; SMN2
SCHEMBL4723847 0.76 HTR6 (0.54) HTR6MEN1P2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003022214-A2 PIPERAZINE AND HOMOPIPERAZINE COMPOUNDS MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-03-20 WO disclosed