SCHEMBL7055846

SCHEMBL7055846

N#Cc1cccc(N2CCN(CCCCNC(=O)c3ccc(Br)cc3)CC2)c1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 14/20 0.73
DRD2 P14416 11/20 0.73
DRD4 P21917 2/20 0.73
KCNH2 Q12809 1/20 0.65
ADRA1A P35348 3/20 0.59
USP2 O75604 1/20 0.53
ALDH1A1 P00352 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MAPT P10636 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058039 0.89 DRD3 (0.79) DRD3DRD2DRD4KCNH2ADRA1A
SCHEMBL7052223 0.85 DRD3 (0.77) DRD3DRD2DRD4ADRA1AUSP2
SCHEMBL24805478 0.85 DRD3 (1.00) DRD3DRD2DRD4
SCHEMBL7052681 0.84 DRD3 (0.67) DRD3DRD2DRD4ADRA1A
SCHEMBL7056313 0.82 DRD3 (0.73) DRD3DRD2DRD4KCNH2ADRA1A
SCHEMBL7057318 0.81 CCR3 (0.54) DRD3DRD2DRD4ALDH1A1
SCHEMBL7056439 0.80 DRD2 (0.76) DRD3DRD2DRD4ADRA1A
SCHEMBL12946337 0.80 DRD3 (0.61) DRD3DRD2DRD4KCNH2ADRA1A
SCHEMBL4536353 0.79 DRD3 (1.00) DRD3DRD2DRD4KCNH2ADRA1A
SCHEMBL7050873 0.78 DRD2 (0.67) DRD3DRD2DRD4KCNH2ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed