SCHEMBL7052223

SCHEMBL7052223

NC(=O)c1cccc(N2CCN(CCCCNC(=O)c3ccc(Br)cc3)CC2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 12/20 0.77
DRD2 P14416 11/20 0.77
ADRA1A P35348 3/20 0.62
DRD4 P21917 2/20 0.59
HTR7 P34969 2/20 0.59
HTR1A P08908 1/20 0.59
HTR2A P28223 1/20 0.59
HTR6 P50406 1/20 0.59
MAPT P10636 1/20 0.58
FAAH O00519 2/20 0.57
USP2 O75604 1/20 0.55
ALDH1A1 P00352 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7055846 0.85 DRD3 (0.73) DRD3DRD2ADRA1ADRD4MAPT
SCHEMBL7056439 0.83 DRD2 (0.76) DRD3DRD2ADRA1ADRD4
SCHEMBL31061220 0.81 DRD3 (0.84) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL7057592 0.81 OPRK1 (0.57) DRD3DRD2DRD4ALDH1A1
SCHEMBL4525601 0.80 HSD17B10 (0.72) DRD3DRD2ADRA1ADRD4HTR1A
SCHEMBL3205704 0.78 HTR7 (0.62) DRD3DRD2HTR7HTR1AHTR2A
SCHEMBL4521840 0.78 DRD4 (0.77) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL7369877 0.77 DRD3 (0.77) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL14006003 0.77 TSHR (0.70) DRD3DRD2DRD4MAPTALDH1A1
SCHEMBL3205692 0.77 HTR7 (0.63) DRD3DRD2HTR7HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed