SCHEMBL7056147

SCHEMBL7056147

CCn1cc(C(=O)NCCc2ccncc2)c(=O)c2cccc(C)c21

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.60
PDE4B Q07343 8/20 0.60
PDE4C Q08493 8/20 0.60
PDE4D Q08499 8/20 0.60
CNR2 P34972 3/20 0.53
RAB9A P51151 2/20 0.49
POLB P06746 1/20 0.49
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
NPY5R Q15761 1/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7051886 0.85 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DCNR2
Hydrochloric Acid SCHEMBL7056139 0.84 PDE4A (0.61) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL7053642 0.84 PDE4A (0.72) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL7057844 0.82 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL7051890 0.81 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL7056821 0.81 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL7055488 0.80 PDE4A (0.77) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL7055652 0.80 ALDH1A1 (0.57) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL6546036 0.80 KMT2A (0.71) PDE4APDE4BPDE4CPDE4DRAB9A
Hydrochloric Acid SCHEMBL7051870 0.79 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0841929-B1 QUINOLONES AND THEIR THERAPEUTIC USE DARWIN DISCOVERY LTD (GB) 2003-05-07 EP claimed