SCHEMBL7067348

SCHEMBL7067348

CCO/C(=C(\C#N)c1ccccc1)c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
ESR1 P03372 1/20 0.39
SIRT3 Q9NTG7 1/20 0.38
MAPT P10636 3/20 0.38
ALDH1A1 P00352 3/20 0.38
KMT2A Q03164 5/20 0.38
MEN1 O00255 4/20 0.38
HPGD P15428 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TP53 P04637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
ALOX12 P18054 1/20 0.36
ELANE P08246 1/20 0.36
AGTR1 P30556 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7067350 1.00 CYP19A1 (0.41) CYP19A1SMN1; SMN2CES2CES1ESR1
SCHEMBL2200157 0.76 SMN1; SMN2 (0.46) SMN1; SMN2MAPTALDH1A1KMT2AMEN1
SCHEMBL8032377 0.75 ELANE (0.43) CYP19A1SMN1; SMN2CES2CES1MAPT
SCHEMBL8032380 0.75 ELANE (0.43) CYP19A1SMN1; SMN2CES2CES1MAPT
SCHEMBL8022876 0.74 CES2 (0.48) SMN1; SMN2CES2CES1ESR1MAPT
SCHEMBL7792871 0.74 SMN1; SMN2 (0.48) SMN1; SMN2MAPTALDH1A1KMT2AMEN1
SCHEMBL13278304 0.73 ALDH1A1 (0.41) SMN1; SMN2MAPTALDH1A1KMT2AMEN1
SCHEMBL27879907 0.71 KMT2A (0.48) SMN1; SMN2MAPTALDH1A1KMT2AMEN1
SCHEMBL9621956 0.71 CES2 (0.42) CYP19A1SMN1; SMN2CES2CES1ESR1
SCHEMBL6396731 0.71 SMN1; SMN2 (0.48) SMN1; SMN2MAPTALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996614-B1 ACRYLONITRILE COMPOUNDS, PROCESS FOR THEIR PRODUCTION AND PESTICIDES CONTAINING THEM ISHIHARA SANGYO KAISHA (JP) 2003-06-11 EP claimed
US-6187944-B1 A PHENYL ACRYLONITRILE COMPOUNDS USEFUL AS ACTIVE INGREDIENTS OF AN INSECTICIDE, A MITICIDE, A NEMATICIDE, A SOIL PESTICIDE, A FUNGICIDE AND A MARINE ANTIFOULING AGENT ISHIHARA SANGYO KAISHA LTD. (JP) 2001-02-13 US claimed
EP-0996614-A1 ACRYLONITRILE COMPOUNDS, PROCESS FOR THEIR PRODUCTION AND PESTICIDES CONTAINING THEM ISHIHARA SANGYO KAISHA, LTD. (JP) 2000-05-03 EP claimed
WO-1998035935-A1 ACRYLONITRILE COMPOUNDS, PROCESS FOR THEIR PRODUCTION AND PESTICIDES CONTAINING THEM ISHIHARA SANGYO KAISHA LTD. (JP) 1998-08-20 WO claimed
EP-0996614-B1 ACRYLONITRILE COMPOUNDS, PROCESS FOR THEIR PRODUCTION AND PESTICIDES CONTAINING THEM ISHIHARA SANGYO KAISHA (JP) 2003-06-11 EP disclosed
US-6187944-B1 A PHENYL ACRYLONITRILE COMPOUNDS USEFUL AS ACTIVE INGREDIENTS OF AN INSECTICIDE, A MITICIDE, A NEMATICIDE, A SOIL PESTICIDE, A FUNGICIDE AND A MARINE ANTIFOULING AGENT ISHIHARA SANGYO KAISHA LTD. (JP) 2001-02-13 US disclosed
EP-0996614-A1 ACRYLONITRILE COMPOUNDS, PROCESS FOR THEIR PRODUCTION AND PESTICIDES CONTAINING THEM ISHIHARA SANGYO KAISHA, LTD. (JP) 2000-05-03 EP disclosed
WO-1998035935-A1 ACRYLONITRILE COMPOUNDS, PROCESS FOR THEIR PRODUCTION AND PESTICIDES CONTAINING THEM ISHIHARA SANGYO KAISHA LTD. (JP) 1998-08-20 WO disclosed