SCHEMBL7070548

SCHEMBL7070548

Cc1nc(-c2ccc(CN3CCN(C(=O)c4ccc(-c5ccccc5)cc4)CC3)cc2)no1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.56
ALDH1A1 P00352 4/20 0.54
MAPT P10636 3/20 0.54
KMT2A Q03164 3/20 0.54
KDM4E B2RXH2 3/20 0.54
LMNA P02545 2/20 0.54
MEN1 O00255 2/20 0.54
RECQL P46063 1/20 0.54
TSHR P16473 2/20 0.54
STAT3 P40763 2/20 0.54
LSS P48449 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HSD17B10 Q99714 1/20 0.54
MAPK1 P28482 1/20 0.54
CHKA P35790 1/20 0.54
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
CYP2D6 P10635 1/20 0.53
KCNH2 Q12809 1/20 0.53
S1PR4 O95977 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074772 0.90 MGLL (0.66) MGLLALDH1A1MAPTKMT2ALMNA
SCHEMBL7071609 0.89 NPC1 (0.65) MGLLALDH1A1MAPTKMT2ALMNA
SCHEMBL7999939 0.85 MGLL (0.52) MGLLKMT2AS1PR4S1PR1S1PR5
SCHEMBL7071582 0.80 LMNA (0.60) MGLLALDH1A1KMT2ALMNAMEN1
SCHEMBL7069980 0.80 TSHR (0.54) ALDH1A1MAPTLMNATSHRLSS
SCHEMBL5928243 0.79 TSHR (0.49) ALDH1A1MAPTKMT2AKDM4ELMNA
SCHEMBL7073717 0.79 TSHR (0.57) MGLLALDH1A1KMT2ALMNARECQL
SCHEMBL12541538 0.79 LSS (0.77) MGLLALDH1A1MAPTKMT2AKDM4E
SCHEMBL5225958 0.79 SMN1; SMN2 (0.59) ALDH1A1MAPTKDM4ELMNATSHR
SCHEMBL7076687 0.79 TSHR (0.59) MGLLALDH1A1MAPTKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed