SCHEMBL7074772

SCHEMBL7074772

Cc1nc(-c2ccc(C(=O)N3CCN(C(=O)c4ccc(-c5ccccc5)cc4)CC3)cc2)no1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.66
POLB P06746 2/20 0.59
HDAC4 P56524 3/20 0.57
HPGD P15428 1/20 0.56
MAPK1 P28482 1/20 0.56
SLC6A7 Q99884 3/20 0.55
HDAC6 Q9UBN7 2/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
MAPT P10636 1/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
FASN P49327 1/20 0.54
PLK1 P53350 1/20 0.53
TSHR P16473 3/20 0.53
ALDH1A1 P00352 3/20 0.53
LMNA P02545 2/20 0.53
NPSR1 Q6W5P4 1/20 0.53
DGAT1 O75907 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7070548 0.90 MGLL (0.56) MGLLMAPK1MAPTMEN1KMT2A
SCHEMBL7071582 0.89 LMNA (0.60) MGLLMEN1KMT2ATSHRALDH1A1
SCHEMBL7076687 0.88 TSHR (0.59) MGLLPOLBHDAC4HPGDHDAC6
SCHEMBL7649408 0.87 DGAT1 (0.58) MGLLPOLBHDAC4MAPTPLK1
SCHEMBL7075122 0.86 LMNA (0.65) MGLLHDAC4TSHRALDH1A1LMNA
SCHEMBL7071696 0.85 ALDH1A1 (0.61) MGLLPOLBHDAC4HDAC6HDAC2
SCHEMBL7075403 0.84 ALDH1A1 (0.57) MGLLPOLBMEN1KMT2AALDH1A1
SCHEMBL7074159 0.84 MGLL (0.55) MGLLPOLBHDAC4MAPK1HDAC6
SCHEMBL3099478 0.84 MGLL (0.55) MGLLHDAC4HDAC6HDAC2HDAC8
SCHEMBL7075196 0.84 MGLL (0.54) MGLLHDAC4MAPK1HDAC6HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed