SCHEMBL7071973

SCHEMBL7071973

CC(C)(C)OC(=O)C(N[C@H]1C=C[C@H](N(C(=O)OC(C)(C)C)C2CCCc3cccnc32)CC1)c1nc2ccccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 20/20 0.44
CHRM2 P08172 1/20 0.39
CYP2D6 P10635 1/20 0.39
DRD2 P14416 1/20 0.39
OPRM1 P35372 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3373807 0.81 SLC40A1 (0.46) CXCR4
SCHEMBL5050922 0.74 CXCR4 (0.50) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL3373810 0.73 CXCR4 (0.68) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL5054117 0.73 CXCR4 (0.38) CXCR4
SCHEMBL4828641 0.72 CXCR4 (0.48) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL3375140 0.72 CXCR4 (0.47) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL5061722 0.71 CXCR4 (0.41) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL3376108 0.69 CXCR4 (0.43) CXCR4
SCHEMBL21651852 0.69 CXCR4 (0.72) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4761001 0.67 CXCR4 (0.67) CXCR4CHRM2CYP2D6DRD2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030220341-A1 Chemokine receptor binding heterocyclic compounds with enhanced efficacy ANORMED, INC. (CA) 2003-11-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030220341-A1 Chemokine receptor binding heterocyclic compounds with enhanced efficacy CCR5, CXCR4, CXCR3 CXCR4 2/4885CHRM2 2757/4885CYP2D6 3057/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.