SCHEMBL7072218

SCHEMBL7072218

Cc1nc(-c2ccc(C(=O)N3CCN(S(=O)(=O)c4c(C)noc4C)CC3)cc2)no1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.53
ATM Q13315 1/20 0.52
HTT P42858 5/20 0.51
HPGD P15428 1/20 0.51
TSHR P16473 2/20 0.49
POLB P06746 1/20 0.49
LMNA P02545 4/20 0.48
MGLL Q99685 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
THRB P10828 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PKM P14618 4/20 0.47
ALDH1A1 P00352 3/20 0.47
CHRM4 P08173 1/20 0.47
USP2 O75604 2/20 0.46
MAPK1 P28482 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7076839 0.85 KMT2A (0.59) POLBLMNAMGLLSMN1; SMN2THRB
SCHEMBL7075196 0.83 MGLL (0.54) TSHRLMNAMGLLTHRBMEN1
SCHEMBL7074432 0.83 HDAC4 (0.47) LMNAMGLLTHRBALDH1A1HDAC4
SCHEMBL7075122 0.83 LMNA (0.65) HTTTSHRLMNAMGLLSMN1; SMN2
SCHEMBL7074222 0.83 LMNA (0.62) HTTLMNAMGLLSMN1; SMN2THRB
SCHEMBL7070540 0.82 TSHR (0.54) SCN9AATMHTTHPGDTSHR
SCHEMBL7071582 0.81 LMNA (0.60) ATMHTTTSHRLMNAMGLL
SCHEMBL7071746 0.81 MEN1 (0.54) HTTPOLBLMNAMGLLSMN1; SMN2
Acetic Acid SCHEMBL27525156 0.81 HTT (0.52) SCN9AATMHTTHPGDTSHR
SCHEMBL7069910 0.81 MGLL (0.52) TSHRLMNAMGLLTHRBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed