SCHEMBL7073367

SCHEMBL7073367

COc1ccc(Oc2c(Br)cc(Br)c(C)c2Br)cc1C(C)C

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
THRB P10828 13/20 0.56
THRA P10827 10/20 0.56
RORC P51449 4/20 0.50
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5283822 0.83 THRB (0.57) THRBTHRARORC
SCHEMBL5041163 0.83 THRB (0.52) THRBTHRARORC
SCHEMBL8893247 0.82 THRB (0.57) THRBTHRARORCCYP2D6
SCHEMBL8892589 0.81 THRB (0.53) THRBTHRARORCCYP2D6
SCHEMBL3886566 0.80 THRB (0.57) THRBTHRARORC
SCHEMBL16496567 0.77 THRB (0.53) THRBTHRARORC
SCHEMBL7071121 0.77 THRB (0.55) THRBTHRARORC
SCHEMBL7076989 0.77 THRB (0.73) THRBTHRARORC
SCHEMBL5618523 0.77 THRB (0.53) THRBTHRARORCCYP2D6
SCHEMBL8064329 0.77 THRB (0.49) THRBTHRARORCCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000008-B1 NOVEL THYROID RECEPTOR LIGANDS AND METHOD KAROBIO AB (SE) 2003-06-25 EP disclosed
US-6465687-B1 SUBSTITUTED 4-HYDROXY-3-ALKYL- OR CYCLOALKYL-PHENOXYBENZENE COMPOUNDS SUCH AS 3,5-DIBROMO-4-(4-HYDROXY-3-ISOPROPYLPHENOXY)BENZOIC ACID, EXPRESSION INHIBITION OF A T3 REGULATED GENE KARO BIO AB (SE) 2002-10-15 US disclosed