SCHEMBL7075345

SCHEMBL7075345

Cc1nc(-c2ccc(C(=O)N3CCN(S(=O)(=O)c4cccs4)CC3)cc2)no1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.56
ALDH1A1 P00352 3/20 0.56
RAB9A P51151 3/20 0.56
PKM P14618 6/20 0.53
MGLL Q99685 1/20 0.49
CA9 Q16790 1/20 0.48
POLB P06746 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
THRB P10828 1/20 0.46
LMNA P02545 3/20 0.46
NPC1 O15118 2/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7075122 0.83 LMNA (0.65) ALDH1A1MGLLHDAC4THRBLMNA
SCHEMBL7075196 0.82 MGLL (0.54) KMT2AALDH1A1MGLLCA9HDAC4
SCHEMBL7071582 0.82 LMNA (0.60) KMT2AALDH1A1MGLLLMNAHTT
SCHEMBL7074222 0.81 LMNA (0.62) KMT2AALDH1A1MGLLTHRBLMNA
SCHEMBL7074799 0.81 MGLL (0.55) KMT2AALDH1A1MGLLHDAC4HDAC2
SCHEMBL7074172 0.80 SMN1; SMN2 (0.56) KMT2AALDH1A1MGLLPOLBTHRB
SCHEMBL7071746 0.80 MEN1 (0.54) KMT2AALDH1A1MGLLCA9POLB
SCHEMBL7072218 0.80 SCN9A (0.53) KMT2AALDH1A1PKMMGLLPOLB
SCHEMBL7076839 0.80 KMT2A (0.59) KMT2AALDH1A1MGLLPOLBHDAC4
SCHEMBL7076931 0.79 MGLL (0.53) KMT2AALDH1A1PKMMGLLHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed