SCHEMBL7076185

SCHEMBL7076185

C=Cc1ccc2cc(OC)ccc2c1.CCN(CC)CC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.44
MAOA P21397 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP2A6 P11509 2/20 0.43
HTR2C P28335 1/20 0.42
NQO2 P16083 2/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
NSD2 O96028 1/20 0.41
S100A4 P26447 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
NOD2 Q9HC29 1/20 0.41
ESR1 P03372 4/20 0.41
AHR P35869 2/20 0.41
TRPA1 O75762 1/20 0.40
RELA Q04206 1/20 0.40
ABL1 P00519 1/20 0.40
TTR P02766 1/20 0.40
CYP1A1 P04798 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29566387 0.88 CYP1A2 (0.54) MAOBCYP1A2CYP2A6HTR2CNQO2
SCHEMBL29566047 0.88 CYP1A2 (0.54) MAOBCYP1A2CYP2A6HTR2CNQO2
SCHEMBL190030 0.88 CYP1A2 (0.54) MAOBCYP1A2CYP2A6HTR2CNQO2
SCHEMBL5673218 0.84 CYP1A2 (0.55) MAOBCYP1A2CYP2A6HTR2CNQO2
SCHEMBL3618006 0.84 CYP1A2 (0.50) MAOBCYP1A2CYP2A6HTR2CNQO2
SCHEMBL3627666 0.84 CYP1A2 (0.50) MAOBCYP1A2CYP2A6HTR2CNQO2
SCHEMBL3625535 0.76 RELA (0.50) CYP1A2MEN1NPC1RAB9AKMT2A
SCHEMBL283100 0.73 TRPA1 (0.39) CYP1A2HTR2CNQO2ESR1AHR
SCHEMBL3629029 0.73 RELA (0.47) CYP1A2MEN1NPC1RAB9AKMT2A
SCHEMBL3624946 0.73 RELA (0.47) CYP1A2MEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0961765-B1 PREPARATION OF CARBOXYLIC COMPOUNDS AND THEIR DERIVATIVES ALBEMARLE CORP (US) 2003-07-09 EP claimed
US-6096920-A LARGE-SCALE PRODUCTION OF CERTAIN AROMATICALLY-SUBSTITUTED ALIPHATIC CARBOXYLIC ACIDS AND THEIR ACID DERIVATIVES ALBEMARLE CORPORATION (US) 2000-08-01 US claimed
EP-0961765-A2 PREPARATION OF CARBOXYLIC COMPOUNDS AND THEIR DERIVATIVES ALBEMARLE CORPORATION (US) 1999-12-08 EP claimed
WO-1998030529-A2 PREPARATION OF CARBOXYLIC COMPOUNDS AND THEIR DERIVATIVES ALBEMARLE CORPORATION (US) 1998-07-16 WO claimed