SCHEMBL7076404

SCHEMBL7076404

COC(=O)c1nc(C)sc1-c1cccc(OCCCI)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HCRTR1 O43613 6/20 0.43
HCRTR2 O43614 5/20 0.43
PKM P14618 2/20 0.40
RCE1 Q9Y256 1/20 0.40
HDAC1 Q13547 7/20 0.39
HDAC2 Q92769 7/20 0.39
HDAC8 Q9BY41 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
GAA P10253 1/20 0.39
VDR P11473 1/20 0.38
MAPT P10636 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7128610 0.90 KDM4E (0.44) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL7160789 0.89 KDM4E (0.44) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL2923794 0.89 POLQ (0.46) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL7160562 0.87 HCRTR1 (0.48) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL7071013 0.86 ALDH1A1 (0.47) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL269345 0.84 KDM4E (0.52) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL2929470 0.83 ALDH1A1 (0.49) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL269910 0.79 KDM4E (0.51) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL2930814 0.79 PIN1 (0.46) HCRTR1HCRTR2HDAC6PPARGPPARA
SCHEMBL270026 0.79 KDM4E (0.53) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003051368-A1 N-AROYL CYCLIC AMINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2003-06-26 WO disclosed