SCHEMBL7076527

SCHEMBL7076527

O=C(NC1CCCCC1)c1c(C[N+]2(C3CCNCC3)CCCCC2)c(-c2ccccc2)nc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 11/20 0.54
TACR2 P21452 9/20 0.54
OPRM1 P35372 6/20 0.54
POLB P06746 1/20 0.47
KCNH2 Q12809 2/20 0.46
CNR1 P21554 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
GAA P10253 2/20 0.42
KMT2A Q03164 1/20 0.42
RAB9A P51151 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
EPHX1 P07099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951612 0.88 TACR3 (0.47) TACR3TACR2OPRM1POLBKCNH2
SCHEMBL7080701 0.88 LMNA (0.50) TACR3TACR2OPRM1KCNH2ALDH1A1
Hydrochloric Acid SCHEMBL7077944 0.87 TACR3 (0.47) TACR3TACR2OPRM1POLBKCNH2
SCHEMBL2372430 0.85 TACR3 (0.50) TACR3TACR2OPRM1POLBKCNH2
SCHEMBL7080543 0.82 TACR3 (0.45) TACR3TACR2OPRM1POLBKCNH2
SCHEMBL6582324 0.82 DHODH (0.42) TACR3TACR2OPRM1POLBKCNH2
SCHEMBL6586109 0.80 TRPV4 (0.43) TACR3TACR2OPRM1POLBKCNH2
SCHEMBL6340547 0.79 TACR3 (0.40) TACR3TACR2OPRM1POLBKCNH2
SCHEMBL7076610 0.79 DHODH (0.48) TACR3TACR2OPRM1POLBKCNH2
SCHEMBL7159967 0.79 DHODH (0.46) TACR3TACR2OPRM1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339691-A1 NOVEL COMPOUNDS GlaxoSmithKline S.p.A. (IT) 2003-09-03 EP disclosed
WO-2002044154-A1 NOVEL COMPOUNDS GLAXOSMITHKLINE SPA (IT) 2002-06-06 WO disclosed