SCHEMBL7076872

SCHEMBL7076872

N=C(N)c1ccc(CCC(=O)N2CCN(S(=O)(=O)c3ccc(-c4ccccc4)cc3)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.55
F13A1 P00488 1/20 0.55
TGM2 P21980 1/20 0.55
TGM1 P22735 1/20 0.55
ALDH1A1 P00352 4/20 0.53
PKM P14618 4/20 0.52
GAA P10253 4/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
LMNA P02545 2/20 0.52
HTT P42858 1/20 0.52
POLB P06746 1/20 0.52
F2 P00734 3/20 0.51
PRSS1 P07477 2/20 0.51
PLG P00747 2/20 0.51
TPSAB1 Q15661 1/20 0.51
TPSD1 Q9BZJ3 1/20 0.51
TPSG1 Q9NRR2 1/20 0.51
MAPK1 P28482 1/20 0.48
HSP90AA1 P07900 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7073640 0.89 PLG (0.56) F13A1TGM2TGM1ALDH1A1PKM
SCHEMBL7075075 0.87 CNR1 (0.56) F13A1TGM2TGM1ALDH1A1PKM
SCHEMBL7076655 0.87 ALDH1A1 (0.55) F13A1TGM2TGM1ALDH1A1PKM
SCHEMBL7073594 0.86 PKM (0.72) ALDH1A1PKMGAASMN1; SMN2LMNA
SCHEMBL7071445 0.83 F10 (0.62) ALDH1A1GAASMN1; SMN2LMNAPOLB
SCHEMBL7074851 0.82 GAA (0.63) ALDH1A1PKMGAALMNAF2
SCHEMBL7074639 0.82 ALDH1A1 (0.55) ALDH1A1PKMGAASMN1; SMN2LMNA
SCHEMBL7074669 0.81 TSHR (0.56) ALDH1A1GAASMN1; SMN2LMNAF2
SCHEMBL7649426 0.81 ALDH1A1 (0.51) ALDH1A1PKMGAASMN1; SMN2LMNA
SCHEMBL17029140 0.81 POLB (0.72) F13A1TGM2TGM1ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed