SCHEMBL7078445

SCHEMBL7078445

O=C1c2cc(O)ccc2CC12C=C1CC=C(O)C=C1C2

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.36
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CES2 O00748 2/20 0.33
ESR1 P03372 4/20 0.32
ESR2 Q92731 4/20 0.32
MAOB P27338 3/20 0.32
MAOA P21397 2/20 0.32
MAPT P10636 1/20 0.31
TNF P01375 1/20 0.30
UGT1A1 P22309 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7070791 0.90 ESR2 (0.38) CA1CA2CA7CA9ESR1
SCHEMBL7074724 0.69 KDM4E (0.30) CA1CA2CA7CA9ESR1
SCHEMBL7078470 0.67 OPRM1 (0.33)
SCHEMBL7075018 0.66 ESR1 (0.46) ESR1ESR2
SCHEMBL19737863 0.66 PBRM1 (0.47) PBRM1CA1CA2CA7CA9
SCHEMBL6794708 0.64 PBRM1 (0.46) PBRM1CA1CA2CA7CA9
SCHEMBL7076088 0.64 SHBG (0.33)
SCHEMBL6794055 0.63 ESR1 (0.44) PBRM1CA1CA2CA7CA9
SCHEMBL7072886 0.62
SCHEMBL17355128 0.60 ESR1 (0.42) PBRM1CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339662-A1 NOVEL ESTROGEN RECEPTOR LIGANDS AND METHODS III KARO BIO AB (SE) 2003-09-03 EP disclosed
WO-2002046134-A1 NOVEL ESTROGEN RECEPTOR LIGANDS AND METHODS III KARO BIO AB (SE) 2002-06-13 WO disclosed