SCHEMBL7078510

SCHEMBL7078510

N=C(N)c1c(O)c2cc(F)ccc2n(CCC2CC2)c1=O

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.52
NR1I2 O75469 1/20 0.52
HIF1A Q16665 1/20 0.43
PLK1 P53350 1/20 0.40
CNR1 P21554 1/20 0.40
CRY1 Q16526 3/20 0.38
CRY2 Q49AN0 3/20 0.38
PER2 O15055 9/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5332751 0.82 ALDH1A1 (0.60) CYP2C9NR1I2HIF1AALDH1A1SMN1; SMN2
SCHEMBL8243641 0.80 HIF1A (0.67) CYP2C9NR1I2HIF1A
SCHEMBL3958416 0.80 CYP2C9 (0.48) CYP2C9NR1I2HIF1APLK1CNR1
SCHEMBL3959350 0.80 CYP2C9 (0.48) CYP2C9NR1I2HIF1APLK1CNR1
SCHEMBL4137380 0.80 CYP2C9 (0.55) CYP2C9NR1I2HIF1APLK1PER2
SCHEMBL5335435 0.79 ALDH1A1 (0.57) CYP2C9NR1I2HIF1AALDH1A1SMN1; SMN2
SCHEMBL5330885 0.79 ALDH1A1 (0.56) CYP2C9NR1I2HIF1ACNR1ALDH1A1
SCHEMBL8247183 0.77 HIF1A (0.62) CYP2C9NR1I2HIF1A
SCHEMBL8245604 0.76 HIF1A (0.61) CYP2C9NR1I2HIF1A
SCHEMBL6689094 0.74 CYP2C9 (0.76) CYP2C9NR1I2PLK1CRY1CRY2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003059356-A2 NOVEL ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2003-07-24 WO claimed
WO-2003059356-A2 NOVEL ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2003-07-24 WO disclosed