SCHEMBL7081206

SCHEMBL7081206

CNc1nc2nc(-c3ccco3)nc-2c[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.42
ADORA1 P30542 9/20 0.42
ADORA3 P0DMS8 8/20 0.42
ADORA2B P29275 6/20 0.42
POLB P06746 2/20 0.42
APAF1 O14727 1/20 0.42
NPC1 O15118 1/20 0.42
NSD2 O96028 1/20 0.42
RAB9A P51151 1/20 0.42
CACNA1B Q00975 1/20 0.42
APBA1 Q02410 1/20 0.42
SAE1 Q9UBE0 1/20 0.42
UBA2 Q9UBT2 1/20 0.42
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 4/20 0.38
HSD17B10 Q99714 3/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7073246 0.81 POLB (0.44) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL7070801 0.78 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL7078373 0.78 RAB9A (0.41) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL6946402 0.78 ALDH1A1 (0.41) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL7077767 0.74 POLB (0.40) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL7078748 0.70 ALDH1A1 (0.46) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL26794368 0.69 POLB (0.58) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL9292249 0.67 PDE10A (0.50) ADORA2AADORA1POLBAPAF1NPC1
SCHEMBL3269949 0.66 KDM4E (0.38) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL8494359 0.65 ALDH1A1 (0.63) ADORA2AADORA1ADORA3ADORA2BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed