SCHEMBL6946402

SCHEMBL6946402

CSc1nc2nc(-c3ccco3)nc-2c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.41
KMT2A Q03164 8/20 0.41
MEN1 O00255 4/20 0.41
KDM4E B2RXH2 4/20 0.41
BLM P54132 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
POLB P06746 5/20 0.41
SAE1 Q9UBE0 2/20 0.41
UBA2 Q9UBT2 2/20 0.41
APAF1 O14727 1/20 0.41
NSD2 O96028 1/20 0.41
CACNA1B Q00975 1/20 0.41
APBA1 Q02410 1/20 0.41
HPGD P15428 9/20 0.40
HSD17B10 Q99714 7/20 0.40
MAPT P10636 4/20 0.40
ALOX15 P16050 3/20 0.40
PTPN7 P35236 2/20 0.40
RECQL P46063 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7073246 0.80 POLB (0.44) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL7081206 0.78 ADORA2A (0.42) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL7070801 0.77 ADORA2A (0.44) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL7078373 0.77 RAB9A (0.41) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL27405338 0.76 POLB (0.47) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL8990531 0.73 ADORA3 (0.45) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL7077767 0.72 POLB (0.40) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL7078748 0.69 ALDH1A1 (0.46) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL26794368 0.68 POLB (0.58) ALDH1A1KMT2AMEN1KDM4EBLM
SCHEMBL9292249 0.66 PDE10A (0.50) ALDH1A1KMT2AMEN1KDM4EBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed