SCHEMBL7081682

SCHEMBL7081682

COC(=O)[C@H](CN)c1ccc(OC)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 1/20 0.46
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 1/20 0.43
ALDH1A1 P00352 2/20 0.43
POLB P06746 1/20 0.43
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
CHRNA7 P36544 1/20 0.41
ACACB O00763 2/20 0.41
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
LMNA P02545 2/20 0.40
NPC1 O15118 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
NR3C1 P04150 1/20 0.39
OXTR P30559 1/20 0.39
PABPC1 P11940 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3861139 0.89 NNMT (0.44) NNMTKMT2AMEN1KDM4EMAPT
SCHEMBL7083560 0.87 NNMT (0.47) NNMTKMT2AMEN1KDM4EMAPT
SCHEMBL7014236 0.87 NNMT (0.47) NNMTKMT2AMEN1KDM4EMAPT
SCHEMBL7009204 0.86 NNMT (0.42) NNMTKMT2AMEN1KDM4EMAPT
SCHEMBL7165235 0.84 NNMT (0.40) NNMTKMT2AMEN1KDM4EMAPT
Trifluoroacetic Acid SCHEMBL17825627 0.81 DPP4 (0.39) NNMTKMT2AMEN1MAPTALDH1A1
SCHEMBL28756577 0.80 NNMT (0.49) NNMTKMT2AMEN1KDM4EMAPT
SCHEMBL3861559 0.78 MAPT (0.48) KDM4EMAPTALDH1A1CHRNA7ACACB
SCHEMBL25180529 0.77 NNMT (0.46) NNMTKMT2AMEN1KDM4EMAPT
SCHEMBL30474590 0.77 NNMT (0.46) NNMTKMT2AMEN1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6646130-B2 Comprises mixtures of alky esters of 3-(6-methoxy-pyridin-3-yl); for inhibiting bone resorption, restenosis, angiogenesis, diabetic retinopathy, macular degeneration, inflammatory arthritis, cancer, and metastasis MERCK & CO., INC. 2003-11-11 US disclosed
US-20030045555-A1 Process to chiral integrin antagonist beta-amino acid intermediate MERCK SHARP & DOHME CORP. 2003-03-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030045555-A1 Process to chiral integrin antagonist beta-amino acid intermediate ITGB1, ITGB3, ITGA1 NNMT 2517/4885KMT2A 3601/4885MEN1 3303/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.