SCHEMBL7082873

SCHEMBL7082873

CNC(=O)OCc1nc(C(C)C)c(Sc2cccc([N+](=O)[O-])c2)n1Cc1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.40
S1PR3 Q99500 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
KDM4E B2RXH2 3/20 0.36
HTT P42858 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
GNRHR P30968 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
ACHE P22303 1/20 0.34
POLB P06746 1/20 0.34
ALDH1A1 P00352 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087594 0.92 CFTR (0.39) CFTRS1PR3CYP1A2CYP3A4KDM4E
SCHEMBL7084592 0.91 CFTR (0.41) CFTRS1PR3CYP1A2CYP3A4KDM4E
SCHEMBL6975011 0.91 CFTR (0.41) CFTRS1PR3CYP1A2CYP3A4KDM4E
SCHEMBL6965963 0.89 TOP2A (0.40) CYP1A2CYP3A4KDM4EHTTMEN1
SCHEMBL7081110 0.88 S1PR3 (0.39) S1PR3KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL7082819 0.88 NPC1 (0.43) KMT2ANPC1RAB9APOLBALDH1A1
SCHEMBL6969486 0.87 LMNA (0.37) HTTMEN1KMT2AGNRHRPOLB
SCHEMBL6973370 0.87 CFTR (0.43) CFTRS1PR3CYP1A2CYP3A4KDM4E
SCHEMBL7081406 0.87 IRAK4 (0.37) CFTRCYP1A2CYP3A4MEN1KMT2A
SCHEMBL6972931 0.87 CFTR (0.44) CFTRS1PR3CYP1A2CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed