SCHEMBL7082819

SCHEMBL7082819

CNC(=O)OCc1nc(C(C)C)c(Sc2cccc(Cl)c2)n1Cc1ccccn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 3/20 0.37
TP53 P04637 3/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
PTGER1 P34995 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
ENPP2 Q13822 1/20 0.34
SLC6A9 P48067 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
POLB P06746 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PPP1CA P62136 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.33
SLC16A3 O15427 1/20 0.33
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6965296 0.93 NPC1 (0.38) NPC1RAB9AMAPTSMN1; SMN2TP53
SCHEMBL7081153 0.91 MAPT (0.39) NPC1RAB9AMAPTSMN1; SMN2TP53
SCHEMBL6965963 0.91 TOP2A (0.40) NPC1RAB9AMAPTSMN1; SMN2TP53
SCHEMBL6973525 0.90 RAB9A (0.35) NPC1RAB9AMAPTSMN1; SMN2TP53
SCHEMBL7081110 0.90 S1PR3 (0.39) NPC1RAB9AMAPTSMN1; SMN2GRIN1
SCHEMBL7081501 0.90 NPC1 (0.38) NPC1RAB9AMAPTSMN1; SMN2TP53
SCHEMBL7082873 0.88 CFTR (0.40) NPC1RAB9AMAPTSMN1; SMN2TDP1
SCHEMBL7084851 0.87 P2RX3 (0.35) TP53RXFP1ENPP2TDP1POLB
SCHEMBL7084180 0.87 S1PR3 (0.39) NPC1RAB9ASMN1; SMN2ENPP2LMNA
SCHEMBL7078929 0.86 TP53 (0.37) RAB9AMAPTSMN1; SMN2TP53RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed