SCHEMBL7083049

SCHEMBL7083049

Cc1cc(C)cc(Sc2c(C(C)C)nc(CCO)n2Cc2cccnc2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.36
LMNA P02545 1/20 0.34
TLR7 Q9NYK1 4/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPT P10636 1/20 0.33
BRD4 O60885 1/20 0.33
GABRA1 P14867 2/20 0.33
GABRA5 P31644 2/20 0.33
ALOX5AP P20292 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
GRIN1 Q05586 2/20 0.32
GRIN2B Q13224 2/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082316 0.94 TLR7 (0.36) SRCLMNATLR7CYP1A2CYP3A4
SCHEMBL6970546 0.92 SRC (0.37) SRCLMNATLR7CYP1A2CYP3A4
SCHEMBL7087528 0.89 SRC (0.35) SRCTLR7MAPTGABRA1GABRA5
SCHEMBL6975018 0.89 GRIN1 (0.38) SRCTLR7ALOX5APHDAC1HDAC8
SCHEMBL7081149 0.89 TLR7 (0.39) SRCTLR7ALOX5APHDAC1HDAC8
SCHEMBL7082502 0.89 BRD4 (0.38) LMNATLR7MAPTBRD4KDM4E
SCHEMBL6972780 0.88 MEN1 (0.33) MEN1KMT2A
SCHEMBL7085996 0.86 ALDH1A1 (0.39) SRCLMNAGABRA1GABRA5GRIN1
SCHEMBL6975548 0.86 GRIN1 (0.38) SRCCYP3A4GRIN1GRIN2B
SCHEMBL6973955 0.86 ALDH1A1 (0.35) LMNATLR7CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed