SCHEMBL6973955

SCHEMBL6973955

Cc1cc(C)cc(Sc2c(C(C)C)nc(CCOC(N)=O)n2Cc2cccnc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
HPGD P15428 2/20 0.35
MEN1 O00255 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
S1PR3 Q99500 3/20 0.35
GABRA1 P14867 3/20 0.35
GABRA5 P31644 3/20 0.35
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973707 0.95 ALDH1A1 (0.34) ALDH1A1KDM4EHPGDMEN1CASP1
SCHEMBL7078695 0.91 CYP1A2 (0.36) ALDH1A1KDM4EHPGDMEN1CASP1
SCHEMBL6966178 0.91 ADRA1D (0.36) ALDH1A1MEN1KMT2AS1PR3GABRA1
SCHEMBL6974966 0.91 GRIN1 (0.36) S1PR3HDAC1HDAC8TLR7
SCHEMBL6974469 0.91 TLR7 (0.36) ALDH1A1KDM4EKMT2AS1PR3GABRA1
SCHEMBL6972473 0.90 LMNA (0.36) ALDH1A1KDM4EHPGDCASP1CASP7
SCHEMBL6964122 0.90 P2RX3 (0.34) ALDH1A1KDM4EHPGDMEN1CASP1
SCHEMBL6973316 0.88 ALDH1A1 (0.39) ALDH1A1MEN1KMT2AGABRA1GABRA5
SCHEMBL7080841 0.88 GRIN1 (0.36) ALDH1A1KMT2AS1PR3LMNA
SCHEMBL6966597 0.86 FKBP1A (0.35) S1PR3GABRA1GABRA5LMNATLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed