SCHEMBL6970546

SCHEMBL6970546

Cc1cc(C)cc(Sc2c(C(C)C)nc(CO)n2Cc2cccnc2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.37
GABRA1 P14867 3/20 0.35
GABRA5 P31644 3/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
BRD4 O60885 1/20 0.34
ALOX5AP P20292 1/20 0.34
TLR7 Q9NYK1 3/20 0.33
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083049 0.92 SRC (0.36) SRCGABRA1GABRA5LMNAMAPT
SCHEMBL7082316 0.90 TLR7 (0.36) SRCGABRA1GABRA5LMNAMAPT
SCHEMBL6969539 0.89 GRIN1 (0.39) SRCALOX5APTLR7GRIN1GRIN2B
SCHEMBL6973652 0.89 SRC (0.37) SRCGABRA1GABRA5MAPTALOX5AP
SCHEMBL7081083 0.89 ALOX5AP (0.37) SRCGABRA1GABRA5LMNAALOX5AP
SCHEMBL6967543 0.88 TDP1 (0.38) LMNAMAPTCYP3A4CYP2C19BRD4
SCHEMBL7083001 0.87 MEN1 (0.34) BRD4KDM4EMEN1ALDH1A1HPGD
SCHEMBL7083464 0.85 GRIN1 (0.39) SRCLMNAMAPTCYP1A2CYP3A4
SCHEMBL6970034 0.85 ALDH1A1 (0.40) SRCGABRA1GABRA5LMNAGRIN1
SCHEMBL7078695 0.85 CYP1A2 (0.36) GABRA1GABRA5LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed