SCHEMBL7083464

SCHEMBL7083464

CC(C)c1nc(CO)n(Cc2cccnc2)c1Sc1cccc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 11/20 0.39
GRIN2B Q13224 11/20 0.39
SRC P12931 1/20 0.35
CYP11B2 P19099 1/20 0.34
KMT2A Q03164 2/20 0.34
CYP3A4 P08684 2/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34
IDO1 P14902 1/20 0.34
CYP17A1 P05093 1/20 0.34
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
ATM Q13315 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975548 0.93 GRIN1 (0.38) GRIN1GRIN2BSRCCYP11B2CYP3A4
SCHEMBL6969539 0.92 GRIN1 (0.39) GRIN1GRIN2BSRCCYP11B2IDO1
SCHEMBL6969811 0.91 GRIN1 (0.37) GRIN1GRIN2BSRCCYP11B2
SCHEMBL6974887 0.90 GRIN1 (0.39) GRIN1GRIN2BSRCCYP11B2CYP3A4
SCHEMBL8109545 0.89 GRIN1 (0.36) GRIN1GRIN2BCYP11B2KMT2ACYP3A4
SCHEMBL6963828 0.89 GRIN1 (0.37) GRIN1GRIN2BSRCCYP11B2KMT2A
SCHEMBL7079895 0.89 GRIN1 (0.38) GRIN1GRIN2BCYP11B2CYP3A4CYP17A1
SCHEMBL6972991 0.89 GRIN1 (0.38) GRIN1GRIN2BCYP11B2
SCHEMBL6961326 0.89 GRIN1 (0.39) GRIN1GRIN2BCYP11B2KMT2AGAA
SCHEMBL6962104 0.89 GRIN1 (0.36) GRIN1GRIN2BSRCCYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed