SCHEMBL6963828

SCHEMBL6963828

CC(C)c1nc(CN=C(N)N)n(Cc2cccnc2)c1Sc1cccc(F)c1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 10/20 0.37
GRIN2B Q13224 10/20 0.37
CYP17A1 P05093 1/20 0.34
CYP3A4 P08684 1/20 0.34
SRC P12931 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
CYP11B2 P19099 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
GRM2 Q14416 1/20 0.32
IDO1 P14902 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081093 0.93 GRIN1 (0.37) GRIN1GRIN2BSRCTLR7CYP11B2
SCHEMBL6973510 0.90 GRIN1 (0.34) GRIN1GRIN2BCYP17A1CYP3A4CYP11B2
SCHEMBL6962312 0.89 HTR3E (0.40) GRIN1GRIN2BSRCTAAR1GAA
SCHEMBL7083464 0.89 GRIN1 (0.39) GRIN1GRIN2BCYP17A1CYP3A4SRC
SCHEMBL6974887 0.89 GRIN1 (0.39) GRIN1GRIN2BCYP17A1CYP3A4SRC
SCHEMBL6969489 0.89 ALDH1A1 (0.37) SRCTLR7
SCHEMBL6975548 0.87 GRIN1 (0.38) GRIN1GRIN2BCYP17A1CYP3A4SRC
SCHEMBL6972991 0.87 GRIN1 (0.38) GRIN1GRIN2BTLR7CYP11B2TAAR1
SCHEMBL6973170 0.87 RECQL (0.43) GRIN1GRIN2BCYP3A4GAAKMT2A
SCHEMBL6969811 0.86 GRIN1 (0.37) GRIN1GRIN2BSRCTLR7CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed