SCHEMBL7079895

SCHEMBL7079895

CC(C)c1nc(CN(C)C)n(Cc2cccnc2)c1Sc1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 11/20 0.38
GRIN2B Q13224 11/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
PKM P14618 1/20 0.34
CYP11B2 P19099 1/20 0.33
CYP17A1 P05093 1/20 0.33
CYP3A4 P08684 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
ROCK2 O75116 1/20 0.33
TLR7 Q9NYK1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082989 0.90 GRIN1 (0.35) GRIN1GRIN2BCYP11B2CYP17A1CYP3A4
SCHEMBL6974922 0.89 POLB (0.41) GRIN1GRIN2BCHRNB2CHRNA4PKM
SCHEMBL6974887 0.89 GRIN1 (0.39) GRIN1GRIN2BCYP11B2CYP17A1CYP3A4
SCHEMBL7083464 0.89 GRIN1 (0.39) GRIN1GRIN2BCYP11B2CYP17A1CYP3A4
SCHEMBL7085922 0.88 CHRNB2 (0.42) CHRNB2CHRNA4TLR7
SCHEMBL6972991 0.87 GRIN1 (0.38) GRIN1GRIN2BCYP11B2TLR7
SCHEMBL6961326 0.87 GRIN1 (0.39) GRIN1GRIN2BCYP11B2
SCHEMBL6975548 0.87 GRIN1 (0.38) GRIN1GRIN2BCYP11B2CYP17A1CYP3A4
SCHEMBL7083193 0.86 GRIN1 (0.38) GRIN1GRIN2BCYP11B2CYP17A1CYP3A4
SCHEMBL6969811 0.85 GRIN1 (0.37) GRIN1GRIN2BCYP11B2TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed