SCHEMBL7083804

SCHEMBL7083804

CC(C)c1nc(COCCO)n(Cc2ccncc2)c1Sc1cccc([N+](=O)[O-])c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.36
PDE4D Q08499 2/20 0.36
PDE4B Q07343 2/20 0.36
POLB P06746 1/20 0.34
MAPT P10636 3/20 0.34
KMT2A Q03164 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP19A1 P11511 3/20 0.33
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 3/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RECQL P46063 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33
SLC2A1 P11166 1/20 0.33
PDE4C Q08493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974930 0.91 RXFP1 (0.36) POLBMAPTKMT2AL3MBTL1CYP19A1
SCHEMBL6967391 0.90 KMT2A (0.35) PDE4APDE4DPDE4BPOLBMAPT
SCHEMBL6974012 0.90 PDE4A (0.38) PDE4APDE4DPDE4BPOLBMAPT
SCHEMBL6969509 0.90 PDE4A (0.34) PDE4APDE4DPDE4BPOLBMAPT
SCHEMBL6963024 0.90 PDE4A (0.39) PDE4APDE4DPDE4BPOLBMAPT
SCHEMBL6970308 0.88 PDE4A (0.37) PDE4APDE4DPDE4BPOLBMAPT
SCHEMBL6971986 0.88 CYP2C9 (0.36) MAPTKMT2AMEN1HPGDCYP2D6
SCHEMBL7084596 0.87 IDO1 (0.33) PDE4DPDE4BMAPTKMT2AALDH1A1
SCHEMBL6969925 0.87 CFTR (0.41) POLBMAPTKMT2AL3MBTL1MEN1
SCHEMBL6968230 0.87 PDE4A (0.36) PDE4APDE4DPDE4BPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed