SCHEMBL7084596

SCHEMBL7084596

CC(C)c1nc(COCCO)n(Cc2ccncc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
PDE4D Q08499 1/20 0.32
PDE4B Q07343 1/20 0.32
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
SLC6A9 P48067 1/20 0.31
GRM5 P41594 1/20 0.31
CSNK2A2 P19784 1/20 0.31
CSNK2B P67870 1/20 0.31
ALDH1A1 P00352 2/20 0.30
MAPT P10636 1/20 0.30
PPP1CA P62136 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
KCNH2 Q12809 1/20 0.30
GSK3B P49841 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970649 0.92 KCNH2 (0.32) GRM5KCNH2
SCHEMBL6972360 0.91 ALDH1A1 (0.37) TDP1GRM5ALDH1A1KMT2ASMN1; SMN2
SCHEMBL7084285 0.90 GRIN1 (0.33) GRM5KMT2A
SCHEMBL8799709 0.90 IDO1 (0.34) IDO1TDP1PDE4DPDE4BGRM5
SCHEMBL6967059 0.90 MAPT (0.33) TDP1ALDH1A1MAPTGSK3B
SCHEMBL6973001 0.89 P2RX3 (0.33) IDO1TDP1ROCK2ROCK1SLC6A9
SCHEMBL6968857 0.88 PIM1 (0.33) IDO1TDP1ROCK2ROCK1SLC6A9
SCHEMBL7087601 0.88 SLC6A9 (0.33) TDP1SLC6A9GRM5ALDH1A1MAPT
SCHEMBL6959029 0.88 IDO1 (0.35) IDO1TDP1PDE4DPDE4BGRM5
SCHEMBL7079909 0.88 IDO1 (0.36) IDO1TDP1PDE4DPDE4BROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed